SCHEMBL22069657

SCHEMBL22069657

O=C(CNCc1ccccc1)Nc1ccc(Oc2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 1.00
LTA4H P09960 1/20 0.70
ALDH1A1 P00352 4/20 0.65
KDM4E B2RXH2 3/20 0.65
SMN1; SMN2 Q16637 2/20 0.65
RNF4 P78317 1/20 0.61
MEN1 O00255 4/20 0.57
KMT2A Q03164 4/20 0.57
GAA P10253 3/20 0.57
POLB P06746 1/20 0.57
HDAC1 Q13547 2/20 0.56
LMNA P02545 2/20 0.56
HPGD P15428 1/20 0.56
MAPT P10636 1/20 0.55
MCHR1 Q99705 2/20 0.55
MCHR2 Q969V1 1/20 0.55
GLA P06280 1/20 0.54
MGLL Q99685 1/20 0.54
HDAC3 O15379 1/20 0.53
HDAC4 P56524 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22069595 0.87 RECQL (0.77) RECQLLTA4HALDH1A1KDM4ESMN1; SMN2
SCHEMBL27852723 0.86 RECQL (0.74) RECQLLTA4HALDH1A1KDM4EMEN1
SCHEMBL22069565 0.86 RECQL (0.75) RECQLLTA4HALDH1A1KDM4ESMN1; SMN2
SCHEMBL6721335 0.86 RECQL (0.75) RECQLLTA4HALDH1A1SMN1; SMN2MEN1
SCHEMBL22069745 0.83 RECQL (0.71) RECQLLTA4HALDH1A1KDM4ESMN1; SMN2
SCHEMBL5316075 0.83 LTA4H (1.00) RECQLLTA4HALDH1A1KDM4ESMN1; SMN2
SCHEMBL8302598 0.82 RECQL (0.70) RECQLLTA4HALDH1A1KDM4ESMN1; SMN2
SCHEMBL5864374 0.82 RECQL (0.69) RECQLALDH1A1KDM4EMEN1KMT2A
SCHEMBL18657627 0.81 RAB9A (0.74) RECQLALDH1A1SMN1; SMN2RNF4MEN1
SCHEMBL22069728 0.81 KDM4E (0.74) RECQLLTA4HALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed