SCHEMBL22071806

SCHEMBL22071806

CCSc1nc2c(cnn2C(C)C)c(=O)[nH]1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.59
ESR1 P03372 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
PDE9A O76083 14/20 0.52
SMN1; SMN2 Q16637 1/20 0.50
ALDH1A1 P00352 1/20 0.49
TSHR P16473 1/20 0.49
KDM4C Q9H3R0 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22042833 0.86 PDE9A (0.52) ESR1PDE9AALDH1A1TSHR
SCHEMBL22042948 0.82 CYP1A2 (0.67) L3MBTL1PDE9ASMN1; SMN2ALDH1A1TSHR
SCHEMBL22042903 0.78 LMNA (0.51) LMNASMN1; SMN2ALDH1A1TSHR
SCHEMBL19342087 0.77 DAPK3 (0.61) L3MBTL1PDE9ATSHR
SCHEMBL22072396 0.76 LMNA (0.57) LMNAESR1L3MBTL1PDE9ASMN1; SMN2
SCHEMBL22042945 0.76 RAB9A (0.52) LMNAL3MBTL1PDE9ASMN1; SMN2ALDH1A1
SCHEMBL15745833 0.76 PDE9A (0.54) PDE9A
SCHEMBL16981646 0.76 PDE9A (0.58) PDE9A
SCHEMBL22071795 0.75 ALDH1A1 (0.82) LMNAESR1L3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL19342102 0.75 MEN1 (0.69) LMNAPDE9AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020116972-A1 COMPOUNDS HAVING PDE9A INHIBITORY ACTIVITY, AND PHARMACEUTICAL USES THEREOF 한국화학연구원 2020-06-11 WO disclosed