SCHEMBL2208

SCHEMBL2208

COC(=O)CNCc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 1/20 0.48
WDR5 P61964 1/20 0.48
FFAR1 O14842 2/20 0.47
AKR1B1 P15121 1/20 0.47
ESR2 Q92731 1/20 0.47
MME P08473 1/20 0.45
PTPN1 P18031 1/20 0.42
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
AR P10275 1/20 0.42
ITGB1 P05556 1/20 0.41
ITGA4 P13612 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
PTPN5 P54829 1/20 0.41
ADAM17 P78536 1/20 0.41
GRIA2 P42262 1/20 0.41
GRIA4 P48058 1/20 0.41
EGLN1 Q9GZT9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1629 0.81 MYC (0.45) MYCWDR5FFAR1AKR1B1ESR2
SCHEMBL2103 0.80 MYC (0.47) MYCWDR5FFAR1AKR1B1ESR2
SCHEMBL2545 0.79 L3MBTL1 (0.47) MYCWDR5FFAR1AKR1B1ESR2
SCHEMBL1997225 0.79 ALDH1A1 (0.51) FFAR1ALDH1A1KDM4ETSHRLMNA
SCHEMBL10057911 0.79 MME (0.45) MYCWDR5FFAR1AKR1B1ESR2
SCHEMBL8239406 0.79 MME (0.45) MYCWDR5FFAR1AKR1B1ESR2
SCHEMBL12851876 0.78 ALDH1A1 (0.47) FFAR1ALDH1A1KDM4EHPGDTSHR
Hydrochloric Acid SCHEMBL2743 0.78 L3MBTL1 (0.49) MYCWDR5FFAR1AKR1B1ESR2
SCHEMBL2226 0.78 MYC (0.46) MYCWDR5FFAR1AKR1B1ESR2
SCHEMBL5346390 0.78 LOXL2 (0.53) ALDH1A1KDM4EKDM4CHPGDEGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965592-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1999-10-12 US disclosed
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed