SCHEMBL22083034

SCHEMBL22083034

CNc1cc(C#N)cc(C2CC2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 1/20 0.35
DRD3 P35462 7/20 0.34
DRD2 P14416 6/20 0.34
SLC6A4 P31645 2/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A3 Q01959 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33
GPR35 Q9HC97 1/20 0.33
CYP2D6 P10635 1/20 0.31
TSHR P16473 1/20 0.31
NFKB1 P19838 1/20 0.31
CASP1 P29466 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TTR P02766 1/20 0.31
ALB P02768 1/20 0.31
CTSS P25774 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28642986 0.82 SLC18A3 (0.36) TSHR
SCHEMBL12326822 0.76 HTR2C (0.38) EGLN2DRD3DRD2CYP2D6TSHR
SCHEMBL25908579 0.73 HTR2C (0.35) DRD3DRD2ALDH1A1MAPTNPSR1
SCHEMBL29672154 0.72 TRPM5 (0.39) EGLN2DRD3DRD2
SCHEMBL1978879 0.72 MEN1 (0.38) EGLN2DRD3DRD2CYP2D6TSHR
SCHEMBL24690097 0.72 EGLN2 (0.37) EGLN2DRD3DRD2SLC6A4CYP2D6
SCHEMBL16954813 0.72 EGLN2 (0.37) EGLN2DRD3DRD2CYP2D6TSHR
SCHEMBL16961551 0.72 EGLN2 (0.37) EGLN2DRD3DRD2CYP2D6TSHR
SCHEMBL16959366 0.72 DRD2 (0.40) EGLN2DRD3DRD2CYP2D6TSHR
SCHEMBL16953765 0.71 EGLN2 (0.35) EGLN2DRD3DRD2GRIA1GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020117877-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE AQUINNAH PHARMACEUTICALS, INC. (US) 2020-06-11 WO disclosed