SCHEMBL22089709

SCHEMBL22089709

Cc1cnc(Cl)nc1-c1ccccc1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 8/20 0.47
MYC P01106 1/20 0.47
LDHA P00338 1/20 0.43
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
GAA P10253 1/20 0.43
KMT2A Q03164 1/20 0.43
HSP90AA1 P07900 1/20 0.42
PDK2 Q15119 1/20 0.42
PDK4 Q16654 1/20 0.42
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 2/20 0.41
USP2 O75604 1/20 0.41
TSHR P16473 1/20 0.41
DHODH Q02127 1/20 0.40
PIN1 Q13526 1/20 0.40
POLB P06746 1/20 0.40
JUN P05412 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30956560 0.86 PDK1 (0.43) PDK1MYCHSP90AA1PDK2PDK4
SCHEMBL22090197 0.86 PDK1 (0.43) PDK1MYCHSP90AA1PDK2PDK4
SCHEMBL30956610 0.85 ALDH1A1 (0.46) MYCRAB9ANPC1KMT2AKDM4E
SCHEMBL30956614 0.85 SLC6A3 (0.50) PDK1KMT2AKDM4EALDH1A1TSHR
SCHEMBL5189312 0.79 CNR1 (0.48) KMT2AKDM4EALDH1A1DHODHPOLB
SCHEMBL22529467 0.78 KMT2A (0.44) PDK1GAAKMT2AHSP90AA1PDK2
SCHEMBL8394975 0.76 JUN (0.55) LDHAGAAKMT2AKDM4EALDH1A1
SCHEMBL30956463 0.76 SLC6A4 (0.41) PDK1RAB9ANPC1KMT2AKDM4E
SCHEMBL25552004 0.75 MBNL1 (0.51) PDK1RAB9ANPC1GAAALDH1A1
SCHEMBL30956550 0.75 SLC6A4 (0.40) PDK1KMT2APDK2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119118999-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl and compositions and methods thereof 凌科药业(杭州)有限公司 2024-12-13 CN disclosed
CN-118955477-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl and compositions and methods thereof 凌科药业(杭州)有限公司 2024-11-15 CN disclosed
CN-118903141-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl and compositions and methods thereof 凌科药业(杭州)有限公司 2024-11-08 CN disclosed
CN-118903142-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl and compositions and methods thereof 凌科药业(杭州)有限公司 2024-11-08 CN disclosed
CN-113227074-B Benzamide derivatives of pyrazolyl-amino-pyrimidinyl and compositions and methods thereof 凌科药业(杭州)有限公司 2024-08-16 CN disclosed
CN-118388457-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl and compositions and methods thereof 凌科药业(杭州)有限公司 2024-07-26 CN disclosed
CN-118290403-A Benzamide derivatives of pyrazolyl-amino-pyrimidinyl and compositions and methods thereof 凌科药业(杭州)有限公司 2024-07-05 CN disclosed
EP-3877381-A1 BENZAMIDES OF PYRAZOLYL-AMINO-PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF Lynk Pharmaceuticals Co. Ltd. (CN) 2021-09-15 EP disclosed
WO-2020119819-A1 BENZAMIDES OF PYRAZOLYL-AMINO-PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF LYNK PHARMACEUTICALS CO. LTD. (CN) 2020-06-18 WO disclosed