SCHEMBL22129202

SCHEMBL22129202

N#Cc1ccc(NCc2ccco2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 14/20 0.54
ALDH1A1 P00352 12/20 0.54
GAA P10253 8/20 0.54
HSD17B10 Q99714 7/20 0.54
HPGD P15428 6/20 0.54
MAPK1 P28482 4/20 0.54
LMNA P02545 3/20 0.54
ALOX15 P16050 2/20 0.54
PKM P14618 1/20 0.54
TSHR P16473 1/20 0.54
NPSR1 Q6W5P4 1/20 0.47
MAPT P10636 6/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
KCNH3 Q9ULD8 2/20 0.45
POLB P06746 2/20 0.45
EED O75530 1/20 0.44
SHMT2 P34897 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
NPC1 O15118 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1391074 0.79 MAPT (0.72) KDM4EALDH1A1GAAHPGDMAPK1
SCHEMBL2805209 0.78 ALDH1A1 (0.68) KDM4EALDH1A1GAAHSD17B10HPGD
SCHEMBL14433848 0.78 RAB9A (0.69) KDM4EALDH1A1GAAHSD17B10HPGD
SCHEMBL9528898 0.78 ALDH1A1 (0.70) KDM4EALDH1A1GAAHPGDMAPK1
SCHEMBL4392903 0.78 KCNH3 (0.51) KDM4EALDH1A1MAPK1NPSR1MAPT
SCHEMBL11792458 0.77 SMN1; SMN2 (0.59) KDM4EALDH1A1GAAHSD17B10HPGD
SCHEMBL456092 0.77 GAA (0.58) KDM4EALDH1A1GAAHSD17B10HPGD
SCHEMBL26644710 0.77 KDM4E (0.58) KDM4EALDH1A1GAAHSD17B10HPGD
SCHEMBL10657204 0.77 ALDH1A1 (0.60) KDM4EALDH1A1GAAHSD17B10HPGD
SCHEMBL15455447 0.77 ALDH1A1 (0.54) KDM4EALDH1A1GAAHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020124500-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 江苏凯迪恩医药科技有限公司 2020-06-25 WO disclosed
WO-2020124500-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 江苏凯迪恩医药科技有限公司 2020-06-25 WO disclosed