SCHEMBL22170

SCHEMBL22170

c1ccc(CSc2nnn[nH]2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 3/20 0.50
ALDH1A1 P00352 2/20 0.47
RAB9A P51151 3/20 0.47
NPC1 O15118 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
HSD17B10 Q99714 1/20 0.44
MAOB P27338 1/20 0.44
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
SCN9A Q15858 1/20 0.43
PKM P14618 1/20 0.43
TSHR P16473 1/20 0.43
GFER P55789 1/20 0.43
MEN1 O00255 1/20 0.43
PPARG P37231 1/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
NCOR2 Q9Y618 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetonitrile SCHEMBL8515909 0.91 ALDH1A1 (0.44) DAOALDH1A1RAB9ANPC1L3MBTL1
SCHEMBL10504274 0.84 CYP1A2 (0.45) DAOALDH1A1RAB9ANPC1L3MBTL1
SCHEMBL10503242 0.82 DAO (0.50) DAOALDH1A1RAB9ANPC1L3MBTL1
SCHEMBL7058887 0.78 NPC1 (0.51) ALDH1A1RAB9ANPC1HSD17B10MAOB
SCHEMBL10369265 0.73 RAB9A (0.49) ALDH1A1RAB9ANPC1HSD17B10SMN1; SMN2
SCHEMBL8438111 0.71 ALDH1A1 (0.60) ALDH1A1RAB9ANPC1HSD17B10MAOB
SCHEMBL452473 0.71 ALDH1A1 (0.35) ALDH1A1L3MBTL1HSD17B10MAOBMAPT
SCHEMBL11636643 0.70 HSD17B10 (0.70) ALDH1A1RAB9ANPC1L3MBTL1HSD17B10
SCHEMBL9199735 0.69 LMNA (0.46) ALDH1A1RAB9ASMN1; SMN2TSHRMEN1
SCHEMBL3293517 0.69 ALDH1A1 (0.34) ALDH1A1HSD17B10MAOBMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2733 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119751529-B Nucleotide dimer, preparation method and application thereof Beijing Xuanjingrui Pharmaceutical Technology Co.,Ltd. (CN) 2026-05-26 CN claimed
US-20260125414-A1 PRODUCTION METHOD OF OLIGONUCLEOTIDE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2026-05-07 US claimed
EP-4658396-A1 BELT REACTOR MANUFACTURING PROCESS FOR OLIGOMER SYNTHESIS Arrowhead Pharmaceuticals, Inc. (US) 2025-12-10 EP claimed
US-12492220-B2 Method for the preparation of oligonucleotides THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2025-12-09 US claimed
US-20250313590-A1 Phosphoramidite morpholino monomers towards synthesis/convergent synthesis of PMO, TMO, their chimera oligos in 5 prime to 3 prime direction INDIAN ASSOCIATION FOR THE CULTIVATION OF SCIENCE (IACS) (IN) 2025-10-09 US claimed
US-20250289843-A1 PROCESS FOR PREPARATION OF TARGETING LIGANDS SIXTH STREETLENDING PARTNERS, AS THE ADMINISTRATIVE AGENT 2025-09-18 US claimed
US-20250236637-A1 GUANINE-RICH OLIGONUCLEOTIDES KUROS US LLC 2025-07-24 US claimed
CN-120157720-A Method for preparing and purifying nucleic acid single strand 南京金斯瑞生物科技有限公司 2025-06-17 CN claimed
EP-4559925-A1 PRODUCTION METHOD OF OLIGONUCLEOTIDE Sumitomo Chemical Company, Limited (JP) 2025-05-28 EP claimed
US-20250145656-A1 METHOD FOR PRODUCING OLIGONUCLEOTIDES NITTO DENKO CORPORATION (JP) 2025-05-08 US claimed
US-20080139797-A1 OLIGONUCLEOTIDES CONTAINING HIGH CONCENTRATIONS OF GUANINE MONOMERS INTEGRATED DNA TECHNOLOGIES, INC. (US) 2008-06-12 US claimed
EP-1912980-A2 OXAZOLIDINONES BEARING ANTIMICROBIAL ACTIVITY COMPOSITION AND METHODS OF PREPARATION Wockhardt Limited (IN) 2008-04-23 EP claimed
US-7339052-B2 Phosphoramidite activator for oligonucleotide synthesis HONEYWELL INTERNATIONAL INC. (US) 2008-03-04 US claimed
EP-1848730-A1 PHOSPHORAMIDUTE ACTIVATOR FOR OLIGONUCLEOTIDE SYNTHESIS Honeywell International, Inc. (US) 2007-10-31 EP claimed
WO-2007041071-A2 OLIGONUCLEOTIDE ANALOGUES INCORPORATING 5-AZA-CYTOSINE THEREIN SUPERGEN, INC. (US) 2007-04-12 WO claimed
WO-2007023507-A2 OXAZOLIDINONES BEARING ANTIMICROBIAL ACTIVITY COMPOSITION AND METHODS OF PREPARATION WOCKHARDT LIMITED (IN) 2007-03-01 WO claimed
WO-2006086186-A1 PHOSPHORAMIDUTE ACTIVATOR FOR OLIGONUCLEOTIDE SYNTHESIS HONEYWELL INTERNATIONAL INC. (US) 2006-08-17 WO claimed
US-20060178509-A1 Phosphoramidite activator for oligonucleotide synthesis SOLSTICE ADVANCED MATERIALS US, INC. 2006-08-10 US claimed
CN-1238346-C Method for producing 1-ethoxyl-5-mercapto-tetrazole HUAFENG CHEMICAL CO LTD NANTON (CN) 2006-01-25 CN claimed
CN-1562980-A Method for producing 1-ethoxyl-5-mercapto-tetrazole HUAFENG CHEMICAL CO LTD NANTON (CN) 2005-01-12 CN claimed