SCHEMBL22199023

SCHEMBL22199023

Cc1ccc(Oc2ccccc2)c(-c2ccccc2)c1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.39
TSHR P16473 1/20 0.39
BRD4 O60885 2/20 0.38
ADORA1 P30542 1/20 0.38
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
RIPK1 Q13546 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
NCOA1 Q15788 1/20 0.36
NCOA3 Q9Y6Q9 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11226020 0.90 KMT2A (0.36) TSHRBRD4CYP1A2MEN1MAPT
SCHEMBL22199028 0.82 SLC6A4 (0.39) LTA4HTSHRBRD4ADORA1CYP1A2
SCHEMBL8335880 0.81 FABP3 (0.43) TSHRMEN1MAPTHPGDMAPK1
SCHEMBL8736795 0.80 LTA4H (0.46) LTA4HTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL22184952 0.80 HTR2A (0.36) LTA4HTSHRADORA1CYP1A2CYP2C9
SCHEMBL11749957 0.79 ALDH1A1 (0.45) LTA4HTSHRBRD4CYP1A2CYP2C9
SCHEMBL17628549 0.79 LTA4H (0.44) LTA4HTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL22199037 0.78 SMN1; SMN2 (0.46) CYP1A2CYP2C9CYP2C19MEN1MAPT
Phosphoric Acid SCHEMBL10790076 0.78 CTNNB1 (0.39) BRD4CYP1A2CYP2C9CYP2C19L3MBTL1
SCHEMBL27757744 0.77 ALDH1A1 (0.52) LTA4HTSHRMEN1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed