SCHEMBL22199028

SCHEMBL22199028

Cc1ccc(Oc2ccccc2)c(-c2ccccc2)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.39
HTR2A P28223 2/20 0.39
TTR P02766 1/20 0.37
LTA4H P09960 2/20 0.37
NTRK1 P04629 1/20 0.37
IGF1R P08069 1/20 0.37
FGFR1 P11362 1/20 0.37
NTRK2 Q16620 1/20 0.37
TSHR P16473 1/20 0.37
ADORA1 P30542 1/20 0.36
BRD4 O60885 1/20 0.36
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22199023 0.82 LTA4H (0.39) SLC6A4TTRLTA4HTSHRADORA1
SCHEMBL22184947 0.79 HTR2A (0.36) SLC6A4HTR2ATTRLTA4HNTRK1
SCHEMBL22198964 0.77 BRD4 (0.39) BRD4CYP1A2MAPTHPGDKMT2A
SCHEMBL11749957 0.77 ALDH1A1 (0.45) SLC6A4LTA4HTSHRBRD4CYP1A2
Phosphoric Acid SCHEMBL10790076 0.76 CTNNB1 (0.39) TTRBRD4CYP1A2CYP2C9CYP2C19
SCHEMBL22199037 0.76 SMN1; SMN2 (0.46) CYP1A2CYP2C9CYP2C19MEN1MAPT
SCHEMBL27757744 0.74 ALDH1A1 (0.52) TTRLTA4HTSHRMEN1MAPT
SCHEMBL11235400 0.74 SLC6A4 (0.42) SLC6A4HTR2ALTA4HTSHRBRD4
SCHEMBL10708885 0.74 FABP4 (0.38) BRD4CYP1A2MAPTHPGDKMT2A
SCHEMBL13545692 0.74 ACHE (0.41) SLC6A4TTRBRD4CYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed