SCHEMBL22216455

SCHEMBL22216455

CCNC(=O)c1cnn(C/C(=C/F)CC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.42
HPGD P15428 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C19 P33261 1/20 0.38
GFER P55789 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KLKB1 P03952 7/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
PDK2 Q15119 1/20 0.35
ACHE P22303 2/20 0.35
HTT P42858 1/20 0.35
KLK1 P06870 1/20 0.35
TYK2 P29597 1/20 0.35
KMT2A Q03164 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PRKAB2 O43741 1/20 0.34
ABL1 P00519 1/20 0.34
CSF1R P07333 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22216339 0.90 KLKB1 (0.41) LMNAHPGDL3MBTL1MAPTCYP2C19
SCHEMBL22216435 0.88 L3MBTL1 (0.39) LMNAHPGDL3MBTL1MAPTCYP2C19
SCHEMBL23907287 0.88 LMNA (0.39) LMNAHPGDL3MBTL1MAPTCYP2C19
SCHEMBL23907289 0.88 LMNA (0.39) LMNAHPGDL3MBTL1MAPTCYP2C19
SCHEMBL22216190 0.86 AOC3 (0.42) LMNAHPGDL3MBTL1MAPTCYP2C19
SCHEMBL28426245 0.85 LMNA (0.37) LMNAHPGDL3MBTL1MAPTCYP2C19
SCHEMBL28426244 0.85 LMNA (0.37) LMNAHPGDL3MBTL1MAPTCYP2C19
SCHEMBL22216433 0.83 L3MBTL1 (0.56) LMNAL3MBTL1MAPTCYP2C19GFER
SCHEMBL23920716 0.83 HPGD (0.40) LMNAHPGDL3MBTL1MAPTCYP2C19
SCHEMBL22207024 0.82 LMNA (0.35) LMNAHPGDL3MBTL1MAPTCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3892621-A1 HALOALLYLAMINE COMPOUNDS AND APPLICATION THEREOF Nanjing Transthera Biosciences Co., Ltd. (CN) 2021-10-13 EP disclosed
WO-2020143763-A1 HALOALLYLAMINE COMPOUNDS AND APPLICATION THEREOF 南京药捷安康生物科技有限公司 2020-07-16 WO disclosed