SCHEMBL222254

SCHEMBL222254

COC(=O)Cc1csc(N)n1

nearest known ligand 0.97

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.64
GABRA5 P31644 1/20 0.64
GABRB2 P47870 1/20 0.64
ALDH1A1 P00352 3/20 0.52
SMN1; SMN2 Q16637 4/20 0.50
RAB9A P51151 4/20 0.50
NPC1 O15118 3/20 0.50
TP53 P04637 1/20 0.50
POLB P06746 1/20 0.50
HPGD P15428 1/20 0.50
HTT P42858 1/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
MAPT P10636 2/20 0.46
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6216313 0.98 HSD17B10 (0.62) HSD17B10GABRA5GABRB2ALDH1A1SMN1; SMN2
SCHEMBL27562636 0.84 GABRA5 (0.66) HSD17B10GABRA5GABRB2ALDH1A1SMN1; SMN2
SCHEMBL10995026 0.83 HSD17B10 (0.60) HSD17B10GABRA5GABRB2ALDH1A1SMN1; SMN2
SCHEMBL27742441 0.83 GABRA5 (0.60) HSD17B10GABRA5GABRB2ALDH1A1SMN1; SMN2
SCHEMBL8445 0.83 MEN1 (0.64) HSD17B10GABRA5GABRB2ALDH1A1SMN1; SMN2
SCHEMBL27527998 0.83 GABRA5 (0.51) HSD17B10GABRA5GABRB2ALDH1A1SMN1; SMN2
SCHEMBL8313903 0.83 GABRA5 (0.64) HSD17B10GABRA5GABRB2ALDH1A1SMN1; SMN2
SCHEMBL12780856 0.82 NOS1 (0.56) HSD17B10GABRA5GABRB2ALDH1A1SMN1; SMN2
SCHEMBL10991421 0.82 GABRA5 (0.58) HSD17B10GABRA5GABRB2ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL1631420 0.82 GABRA5 (0.50) HSD17B10GABRA5GABRB2ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 245 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101362735-B Preparation method of ethyl 2-[[(bezyloxy)carbonyl]amido]-4-thiazolyl acetate SHANDONG JINCHENG PHARMACEUTICAL & CHEMICALS CO LTD 2011-01-05 CN claimed
EP-3717459-B1 COMPOUNDS STEP PHARMA S A S (FR) 2026-01-21 EP disclosed
EP-4667054-A2 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY Novartis AG (CH) 2025-12-24 EP disclosed
US-12503466-B2 Aminothiazole compounds as inhibitors of CTPS1 STEP PHARMA S.A.S. (FR) 2025-12-23 US disclosed
EP-3880660-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2025-07-02 EP disclosed
WO-2025048759-A1 BENZIMIDAZOLE DERIVATIVES AS MPGES-1 INHIBITORS ICOSYN THERAPEUTICS SAGLIK TEKNOLOJILERI ANONIM SIRKETI (TR) 2025-03-06 WO disclosed
WO-2024140653-A1 SELECTIVE CDK12/13 INHIBITOR AND APPLICATION THEREOF 南京圣和药业股份有限公司 2024-07-04 WO disclosed
CN-118255746-A Selective CDK12/13 inhibitors and uses thereof 南京圣和药业股份有限公司 2024-06-28 CN disclosed
US-20240010645-A1 Aminothiazole Compounds as Inhibitors of CTPS1 STEP PHARMA S.A.S. (FR) 2024-01-11 US disclosed
EP-4275759-A2 QUINOLINE DERIVATIVES AS CHROMOBOX (CBX) PROTEIN INHIBITORS FOR TREATING CANCER Dana-Farber Cancer Institute, Inc. (US) 2023-11-15 EP disclosed
US-4782147-A ANTIBIOTIC TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-11-01 US disclosed
EP-0053816-B1 1-SULFO-2-OXOAZETIDINE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1988-05-04 EP disclosed
US-4675397-A MICROBIOCIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1987-06-23 US disclosed
US-4665067-A BACTERICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1987-05-12 US disclosed
US-4560765-A USING 183-THIAZOL-4-YL GLYOXYLIC ACID AS INTERMEDIATE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1985-12-24 US disclosed
US-4550105-A BETA-LACTAMASE INHIBITORS, ANTIBIOTICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1985-10-29 US disclosed
US-4500716-A Intermediate products for the preparation of Z-cephalosporins BAYER AKTIENGESELLSCHAFT (DE) 1985-02-19 US disclosed
EP-0093376-A2 1-Sulfo-2-azetidinone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1983-11-09 EP disclosed
EP-0053816-A1 1-Sulfo-2-oxoazetidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1982-06-16 EP disclosed
US-4303655-A MICROBIOCIDES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-12-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12503466-B2 Aminothiazole compounds as inhibitors of CTPS1 CTPS1, CTPS2, TBXAS1 HSD17B10 2038/4885GABRA5 4137/4885GABRB2 2961/4885
US-20240010645-A1 Aminothiazole Compounds as Inhibitors of CTPS1 CTPS1, CTPS2, TBXAS1 HSD17B10 2038/4885GABRA5 4137/4885GABRB2 2961/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.