SCHEMBL2222899

SCHEMBL2222899

Cc1cc(-c2nc3cnc(Oc4ccc(Cl)cc4F)nc3o2)cc(C)c1[O]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.51
CYP3A4 P08684 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
HPGD P15428 2/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HSD17B10 Q99714 1/20 0.37
GRIN2B Q13224 1/20 0.35
PTGS2 P35354 4/20 0.35
PTGS1 P23219 1/20 0.35
ANO1 Q5XXA6 1/20 0.34
APP P05067 2/20 0.34
S1PR4 O95977 1/20 0.34
PPARG P37231 1/20 0.34
CETP P11597 1/20 0.33
FFAR1 O14842 1/20 0.33
PPARD Q03181 1/20 0.33
PPARA Q07869 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2222588 0.93 S1PR1 (0.52) S1PR1CYP3A4CYP1A2CYP2C19HPGD
SCHEMBL2222292 0.90 S1PR1 (0.44) S1PR1
SCHEMBL2222071 0.90 S1PR1 (0.44) S1PR1HPGDTP53MAPTHSD17B10
SCHEMBL2224286 0.89 S1PR1 (0.54) S1PR1CYP3A4CYP1A2CYP2C19HPGD
SCHEMBL2222186 0.88 S1PR1 (0.48) S1PR1CYP3A4CYP1A2HPGDTP53
SCHEMBL2224913 0.86 S1PR1 (0.47) S1PR1CYP3A4CYP1A2CYP2C19HPGD
SCHEMBL2223727 0.86 S1PR1 (0.47) S1PR1HPGDTP53MAPTHSD17B10
SCHEMBL2223599 0.86 S1PR1 (0.47) S1PR1TP53MAPTAPPCETP
SCHEMBL14797056 0.85 S1PR1 (0.73) S1PR1HPGDTP53MAPTNPSR1
SCHEMBL2222853 0.84 S1PR1 (0.58) S1PR1CYP3A4CYP1A2CYP2C19HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523962-A1 CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI (FR) 2012-11-21 EP disclosed
WO-2011086079-A1 CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI-AVENTIS (FR) 2011-07-21 WO disclosed