SCHEMBL2228748

SCHEMBL2228748

CN=C(c1c(NCC2CC2)nc2ccccn2c1=O)C1CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
HPGD P15428 3/20 0.38
ALOX15 P16050 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KDM4E B2RXH2 4/20 0.37
LMNA P02545 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
THRB P10828 1/20 0.36
TP53 P04637 1/20 0.36
VCP P55072 2/20 0.36
RXFP1 Q9HBX9 4/20 0.36
RAB9A P51151 3/20 0.36
GLA P06280 3/20 0.35
GAA P10253 3/20 0.35
CASP1 P29466 2/20 0.35
CASP7 P55210 2/20 0.35
HSD17B10 Q99714 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2228484 0.76 MAPT (0.44) ALDH1A1HPGDALOX15NPSR1KDM4E
SCHEMBL12517668 0.73 ALDH1A1 (0.59) ALDH1A1HPGDALOX15NPSR1KDM4E
SCHEMBL13651125 0.64 ALDH1A1 (0.55) ALDH1A1HPGDALOX15KDM4ERXFP1
SCHEMBL20673899 0.63 PDE10A (0.41) KDM4EVCPADORA2A
SCHEMBL21958603 0.63 PDE10A (0.39) ALDH1A1KDM4EL3MBTL1GAACYP2D6
SCHEMBL2219841 0.62 KMT2A (0.48) ALDH1A1HPGDKDM4ETHRBTP53
SCHEMBL13651130 0.62 DDX3X (0.49) ALDH1A1HPGDALOX15NPSR1KDM4E
SCHEMBL23937735 0.61 HTR4 (0.50) CYP2D6
SCHEMBL15887206 0.61 HPGD (0.60) ALDH1A1HPGDALOX15NPSR1KDM4E
SCHEMBL14552917 0.60 ALDH1A1 (0.63) ALDH1A1HPGDALOX15NPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011089457-A1 NOVEL MEDICINAL COMPOUNDS URATIM GYÁRTÓ KORLÁTOLT FELELŐSSÉGŰ TÁRSASÁG (HU) 2011-07-28 WO claimed
WO-2011089457-A1 NOVEL MEDICINAL COMPOUNDS URATIM GYÁRTÓ KORLÁTOLT FELELŐSSÉGŰ TÁRSASÁG (HU) 2011-07-28 WO disclosed