SCHEMBL22293268

SCHEMBL22293268

Cc1sc(N(CCC2CCCC2)Cc2ccccc2)nc1C=O

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTR2B P41595 1/20 0.35
ACHE P22303 4/20 0.34
SLC6A4 P31645 2/20 0.34
BCHE P06276 2/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
PPARD Q03181 2/20 0.33
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22292917 0.90 ALDH1A1 (0.36) KDM4EALDH1A1HTR2BACHEPPARD
SCHEMBL22293305 0.90 CNR1 (0.36) KDM4EALDH1A1ACHEBCHEPPARD
SCHEMBL22293302 0.88 NR1D1 (0.37) ALDH1A1SLC6A4
SCHEMBL22293291 0.88 KDM4E (0.37) KDM4EALDH1A1HTR2BOPRM1OPRD1
SCHEMBL22293272 0.81 ALDH1A1 (0.39) KDM4EALDH1A1HTR2BSLC6A4
SCHEMBL22293282 0.79 HPGD (0.35) BCHE
SCHEMBL22293004 0.77 KDM4E (0.41) KDM4EALDH1A1HTR2B
SCHEMBL22292961 0.77 KDM4E (0.43) KDM4EALDH1A1HTR2BPPARDSIGMAR1
SCHEMBL18975162 0.76 LPAR1 (0.40) ALDH1A1HTR2BACHESLC6A4BCHE
SCHEMBL18974645 0.75 LPAR1 (0.40) ALDH1A1HTR2BACHESLC6A4BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3388425-B1 AMINOAZOLE DERIVATIVE TEIJIN PHARMA LTD (JP) 2020-08-05 EP disclosed