SCHEMBL22293291

SCHEMBL22293291

Cc1sc(N(Cc2ccccc2)CC2CCCCCC2)nc1C=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
HTR2B P41595 1/20 0.36
ATM Q13315 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
G6PC1 P35575 1/20 0.34
USP2 O75604 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
PKM P14618 1/20 0.34
MAPK1 P28482 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
LPAR1 Q92633 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22293268 0.88 KDM4E (0.36) KDM4EALDH1A1OPRM1OPRD1OPRK1
SCHEMBL22293272 0.82 ALDH1A1 (0.39) KDM4EALDH1A1HTR2BG6PC1USP2
SCHEMBL22293305 0.80 CNR1 (0.36) KDM4EALDH1A1NPC1RAB9ACNR1
SCHEMBL22292917 0.78 ALDH1A1 (0.36) KDM4EALDH1A1HTR2BNPC1RAB9A
SCHEMBL22293302 0.78 NR1D1 (0.37) ALDH1A1ATMNPC1RAB9AMAPK1
SCHEMBL22293004 0.78 KDM4E (0.41) KDM4EALDH1A1HTR2BG6PC1RAB9A
SCHEMBL22293189 0.76 CYP19A1 (0.33) OPRM1OPRD1OPRK1CNR2
SCHEMBL22292920 0.75 KDM4E (0.44) KDM4EALDH1A1
SCHEMBL18974921 0.75 CMKLR1 (0.41) ALDH1A1ATMHDAC1HDAC6MAPK1
SCHEMBL22293027 0.74 ALDH1A1 (0.42) KDM4EALDH1A1HTR2BHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3388425-B1 AMINOAZOLE DERIVATIVE TEIJIN PHARMA LTD (JP) 2020-08-05 EP disclosed