SCHEMBL22309042

SCHEMBL22309042

O=C(c1ccc(I)cc1)C1(c2ccc(I)cc2)OCCO1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.41
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
PHGDH O43175 1/20 0.37
PTPN2 P17706 2/20 0.37
PTPN1 P18031 2/20 0.37
GSK3B P49841 1/20 0.36
RXRA P19793 2/20 0.33
RXRB P28702 2/20 0.33
CYP26A1 O43174 1/20 0.33
CYP26B1 Q9NR63 1/20 0.33
AKR1C3 P42330 1/20 0.32
HIF1A Q16665 2/20 0.31
EPAS1 Q99814 2/20 0.31
RXRG P48443 1/20 0.31
AVPR2 P30518 1/20 0.31
OXTR P30559 1/20 0.31
AVPR1A P37288 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18790751 0.93 TPMT (0.38) TPMTCA1CA2PHGDHPTPN2
SCHEMBL18790764 0.92 POLB (0.38) TPMTCA1CA2PHGDHRXRA
SCHEMBL18790761 0.86 POLB (0.36) TPMTCA1CA2PHGDHRXRA
SCHEMBL22309040 0.83 TPMT (0.36) TPMTCA1CA2PHGDHPTPN2
SCHEMBL11486312 0.82 CES2 (0.42) CA1CA2PHGDHAKR1C3POLB
SCHEMBL18790832 0.82 ALDH1A1 (0.42) RXRARXRBRXRGPOLB
SCHEMBL18790464 0.79 POLB (0.35) TPMTCA1CA2RXRAPOLB
SCHEMBL1551316 0.78 LMNA (0.40) CA1CA2POLB
SCHEMBL22309043 0.77 TPMT (0.39) TPMTCA1CA2PHGDHPTPN2
SCHEMBL11495372 0.76 POLB (0.40) RXRAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3365318-B1 BENZYL MONOKETALS AND USE THEREOF MERCK PATENT GMBH (DE) 2021-01-06 EP disclosed
US-20200247916-A1 BENZIL MONOKETALS AND THE USE THEREOF MERCK PATENT GMBH (DE) 2020-08-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200247916-A1 BENZIL MONOKETALS AND THE USE THEREOF BCKDK, PKLR, BPHL TPMT 867/4885CA1 3127/4885CA2 3368/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.