SCHEMBL2233914

SCHEMBL2233914

CCCC/C(=C\C(=O)O)c1cc(Cl)c(Oc2ccc(OCc3ccc(C)cc3)cn2)cc1C

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACACB O00763 4/20 0.41
PSEN1 P49768 9/20 0.38
ALOX5 P09917 7/20 0.38
PPARG P37231 6/20 0.38
PTGES O14684 4/20 0.38
GRM2 Q14416 1/20 0.37
CYSLTR1 Q9Y271 1/20 0.37
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
ACACA Q13085 2/20 0.36
MAOB P27338 1/20 0.36
PARP10 Q53GL7 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2231811 0.91 ACACB (0.39) ACACBPSEN1ALOX5PPARGPTGES
SCHEMBL2235542 0.87 NR4A2 (0.41) ACACBMAOB
SCHEMBL2233918 0.83 PSEN1 (0.51) PSEN1ALOX5PPARGPTGES
SCHEMBL2231990 0.82 RAB9A (0.38) ACACBPSEN1ALOX5PPARGPTGES
SCHEMBL2233299 0.79 PTGER3 (0.42) ACACBPPARGACACAMAOB
SCHEMBL2233287 0.79 PTGER3 (0.42) ACACBPPARGACACAMAOB
SCHEMBL2233912 0.79 ACACB (0.41) ACACBPSEN1ALOX5PPARGPTGES
SCHEMBL2231815 0.78 PSEN1 (0.51) PSEN1ALOX5PPARGPTGES
SCHEMBL2231791 0.77 PPARG (0.40) ACACBPSEN1ALOX5PPARGPTGES
SCHEMBL2233200 0.77 ALOX5 (0.35) ACACBALOX5PPARGCYP4F2CYP4A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011093524-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-08-04 WO disclosed