SCHEMBL22336151

SCHEMBL22336151

COc1cc(N2CCN(C)CC2)c2oc(CN=O)cc2c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 4/20 0.38
SLC22A12 Q96S37 2/20 0.35
HRH4 Q9H3N8 1/20 0.35
DRD2 P14416 2/20 0.35
DRD3 P35462 2/20 0.35
HTR1A P08908 2/20 0.34
TSHR P16473 2/20 0.34
DRD4 P21917 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
KDM4E B2RXH2 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
HTR1B P28222 2/20 0.34
ELANE P08246 1/20 0.34
LMNA P02545 1/20 0.33
HTR1D P28221 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21225965 0.85 CCR4 (0.38) CCR4SLC22A12HRH4DRD2DRD3
SCHEMBL16623287 0.78 SLC22A12 (0.40) SLC22A12KDM4EELANELMNA
SCHEMBL16623261 0.77 SLC22A12 (0.40) SLC22A12TSHRKDM4EKMT2AMEN1
SCHEMBL21230519 0.74 JAK2 (0.37) SLC22A12KDM4EKMT2A
SCHEMBL21224437 0.72 PRKDC (0.41) SLC22A12TSHRKDM4EKMT2AMEN1
SCHEMBL22336290 0.72 SLC22A12 (0.36) SLC22A12
SCHEMBL21224535 0.71 SLC22A12 (0.36) SLC22A12KDM4E
SCHEMBL22336249 0.68 ALDH1A1 (0.36) SLC22A12TSHRKDM4EKMT2AMEN1
SCHEMBL16623281 0.67 CYP2A6 (0.51) KDM4E
SCHEMBL26244659 0.67 KDM4E (0.39) DRD2DRD3HTR1ADRD4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019152955-A9 SMALL MOLECULE DRUG CONJUGATES OF GEMCITABINE MONOPHOSPHATE EVERETT STEVEN ALBERT (US) 2020-08-13 WO disclosed