SCHEMBL22336249

SCHEMBL22336249

COc1cc(N(C)c2ccccc2)c2oc(CN=O)cc2c1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 2/20 0.36
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SLC22A12 Q96S37 2/20 0.35
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.32
TSHR P16473 1/20 0.32
KMT2A Q03164 1/20 0.32
CSF1R P07333 2/20 0.32
ACHE P22303 2/20 0.31
MTNR1A P48039 2/20 0.31
MTNR1B P49286 2/20 0.31
GPR55 Q9Y2T6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21226532 0.84 SLC22A12 (0.37) ALDH1A1HPGDKDM4ELMNANPSR1
SCHEMBL16623287 0.76 SLC22A12 (0.40) ALDH1A1HPGDKDM4ELMNAHSD17B10
SCHEMBL16623261 0.74 SLC22A12 (0.40) ALDH1A1HPGDKDM4ELMNAHSD17B10
SCHEMBL22336290 0.69 SLC22A12 (0.36) SLC22A12
SCHEMBL26244653 0.68 HSP90AA1 (0.33) MEN1TSHRKMT2A
SCHEMBL26244657 0.68 MAOB (0.34) KDM4ETP53SMN1; SMN2MEN1TSHR
SCHEMBL22336151 0.68 CCR4 (0.38) KDM4ELMNASLC22A12MEN1TSHR
SCHEMBL16623281 0.67 CYP2A6 (0.51) ALDH1A1HPGDKDM4ESMN1; SMN2GPR55
SCHEMBL21224539 0.66 SLC22A12 (0.40) KDM4ESLC22A12
SCHEMBL5608400 0.62 MTNR1A (0.46) ALDH1A1CYP3A4MEN1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019152955-A9 SMALL MOLECULE DRUG CONJUGATES OF GEMCITABINE MONOPHOSPHATE EVERETT STEVEN ALBERT (US) 2020-08-13 WO disclosed