SCHEMBL22336337

SCHEMBL22336337

COc1cc(Br)c(O)c(C(C)O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.41
PTGS2 P35354 1/20 0.41
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
ADRA2A P08913 2/20 0.38
ADRA1A P35348 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
ALDH1A1 P00352 1/20 0.37
LCK P06239 1/20 0.37
PRKACA P17612 1/20 0.37
PRKACG P22612 1/20 0.37
PRKACB P22694 1/20 0.37
MEN1 O00255 1/20 0.37
MAPK1 P28482 1/20 0.37
BLM P54132 1/20 0.37
KMT2A Q03164 1/20 0.37
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
THRA P10827 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6796164 0.81 ADRA2A (0.49) ADRA2AADRA1ACYP3A4CYP2D6MEN1
SCHEMBL14691495 0.81 ADRA2A (0.49) ADRA2AADRA1ACYP3A4CYP2D6MEN1
SCHEMBL1119249 0.79 ALOX5 (0.54) ALOX5PTGS2CA1CA2CYP3A4
SCHEMBL4136739 0.78 GABRA1 (0.56) CA1CA2CYP3A4CYP2D6ALDH1A1
SCHEMBL21526723 0.76 ADRA2A (0.44) ADRA2AADRA1ACYP2D6MEN1MAPK1
SCHEMBL6446902 0.75 LCK (0.40) ALOX5PTGS2CA1CA2CYP3A4
SCHEMBL22897820 0.74 ADRA2A (0.46) CA1CA2ADRA2AADRA1ACYP3A4
SCHEMBL6795750 0.74 ADRA2A (0.46) CA1CA2ADRA2AADRA1ACYP3A4
SCHEMBL2978694 0.74 GABRA1 (0.52) CA1CA2CYP3A4ALDH1A1MEN1
SCHEMBL25912511 0.74 KDM4E (0.49) CA1CA2ALDH1A1KMT2ATHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019152955-A9 SMALL MOLECULE DRUG CONJUGATES OF GEMCITABINE MONOPHOSPHATE EVERETT STEVEN ALBERT (US) 2020-08-13 WO disclosed