SCHEMBL2234193

SCHEMBL2234193

COCCN1C(=O)C(O)=C(C(=O)c2ccc(C)cc2)C1c1ccc(C(C)C)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ANXA2 P07355 5/20 0.67
S100A10 P60903 5/20 0.67
ALDH1A1 P00352 2/20 0.56
KDM4E B2RXH2 2/20 0.56
HPGD P15428 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
CYP2C9 P11712 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
TP53 P04637 2/20 0.53
MAPT P10636 1/20 0.53
MDM2 Q00987 1/20 0.48
FPR1 P21462 3/20 0.46
HTT P42858 1/20 0.46
HIF1A Q16665 1/20 0.46
ALOX15 P16050 3/20 0.46
RXFP1 Q9HBX9 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
USP2 O75604 1/20 0.44
TSHR P16473 1/20 0.44
MALT1 Q9UDY8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2233839 0.94 ANXA2 (0.68) ANXA2S100A10ALDH1A1KDM4EHPGD
SCHEMBL2232974 0.84 ANXA2 (0.65) ANXA2S100A10ALDH1A1MALT1
SCHEMBL681885 0.82 ALDH1A1 (0.53) ANXA2S100A10ALDH1A1KDM4EHPGD
SCHEMBL2303389 0.82 ANXA2 (0.66) ANXA2S100A10ALDH1A1KDM4ETDP1
SCHEMBL2235370 0.81 ANXA2 (0.53) ANXA2S100A10ALDH1A1KDM4ETDP1
SCHEMBL12668752 0.79 PPARG (0.57) ALDH1A1KDM4EMAPTALOX15RXFP1
SCHEMBL2236184 0.77 ANXA2 (0.55) ANXA2S100A10HPGDTDP1CYP2C9
SCHEMBL2232358 0.76 CCR1 (0.59) ANXA2S100A10ALDH1A1KDM4EHPGD
SCHEMBL13927439 0.75 ALDH1A1 (0.52) ANXA2S100A10ALDH1A1KDM4EHPGD
SCHEMBL2234993 0.75 ANXA2 (0.65) ANXA2S100A10ALDH1A1KDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011092505-A1 S100 PROTEIN BINDING INTERACTION INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2011-08-04 WO claimed
WO-2011092505-A1 S100 PROTEIN BINDING INTERACTION INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2011-08-04 WO disclosed