SCHEMBL22355669

SCHEMBL22355669

COc1ccc2c(c1)N(C)C1(CCN(c3ccc(/C(C=N)=C/N)cc3)C1=O)C2

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.32
OPRK1 P41145 1/20 0.32
OPRL1 P41146 1/20 0.32
KYAT1 Q16773 1/20 0.32
KYAT3 Q6YP21 1/20 0.32
AADAT Q8N5Z0 1/20 0.32
BACE1 P56817 1/20 0.32
ITGB3 P05106 5/20 0.31
ITGA2B P08514 5/20 0.31
ALDH1A1 P00352 2/20 0.31
TP53 P04637 2/20 0.31
ALOX15 P16050 2/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
MAPK1 P28482 1/20 0.31
KDM4E B2RXH2 2/20 0.30
MAPT P10636 2/20 0.30
LIPE Q05469 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22355671 0.83 ITGB3 (0.37) ITGB3ITGA2BLIPE
SCHEMBL29443013 0.81 ROCK2 (0.40) OPRM1OPRK1OPRL1BACE1ALDH1A1
SCHEMBL21490353 0.81 ROCK2 (0.40) OPRM1OPRK1OPRL1BACE1ALDH1A1
SCHEMBL22355681 0.77 PPIB (0.37) ITGB3ITGA2BTP53HPGDKDM4E
SCHEMBL22355668 0.77 ROCK2 (0.42) ALDH1A1ALOX15GAAKDM4EMAPT
SCHEMBL29442948 0.75 ROCK2 (0.48)
SCHEMBL21490346 0.75 ROCK2 (0.48)
SCHEMBL24742760 0.72 L3MBTL1 (0.48) ITGB3ITGA2BALDH1A1TP53HPGD
SCHEMBL22355673 0.71 ITGB3 (0.38) ITGB3ITGA2BLIPE
SCHEMBL22355757 0.71 ITGB3 (0.41) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3481817-B1 SPIROLACTAMS AS INHIBITORS OF ROCK BRISTOL MYERS SQUIBB CO (US) 2020-08-19 EP disclosed