SCHEMBL22355671

SCHEMBL22355671

COc1ccc2c(c1)CC1(CCN(c3ccc(/C(C=N)=C/N)cc3)C1=O)C2

nearest known ligand 0.37

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 12/20 0.37
ITGA2B P08514 12/20 0.37
LIPE Q05469 7/20 0.37
OTUD7B Q6GQQ9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22355757 0.86 ITGB3 (0.41) ITGB3ITGA2B
SCHEMBL22355673 0.86 ITGB3 (0.38) ITGB3ITGA2BLIPE
SCHEMBL22355681 0.83 PPIB (0.37) ITGB3ITGA2B
SCHEMBL22355669 0.83 OPRM1 (0.32) ITGB3ITGA2BLIPE
SCHEMBL22355668 0.83 ROCK2 (0.42) LIPEOTUD7B
SCHEMBL24742760 0.80 L3MBTL1 (0.48) ITGB3ITGA2B
SCHEMBL21490362 0.80 ROCK2 (0.44) LIPEOTUD7B
SCHEMBL29443020 0.80 ROCK2 (0.44) LIPEOTUD7B
SCHEMBL22355670 0.79 OTUD7B (0.32) OTUD7B
SCHEMBL24743239 0.79 L3MBTL1 (0.44) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3481817-B1 SPIROLACTAMS AS INHIBITORS OF ROCK BRISTOL MYERS SQUIBB CO (US) 2020-08-19 EP disclosed