SCHEMBL22365602

SCHEMBL22365602

C=CC[C@@]1(Cc2ccccc2)CNCCN1C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
STS P08842 1/20 0.35
MAPK1 P28482 1/20 0.35
GPR119 Q8TDV5 3/20 0.35
ACHE P22303 2/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
KDM4E B2RXH2 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4321471 0.90 STS (0.39) OPRD1OPRK1STSMAPK1GPR119
SCHEMBL24596421 0.81
SCHEMBL22147583 0.80 MAPK1 (0.40) OPRD1OPRK1STSMAPK1GPR119
SCHEMBL22148053 0.78 HCRTR2 (0.33) MEN1KMT2AKDM4E
SCHEMBL27573516 0.76 L3MBTL1 (0.43) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL4394294 0.74 CTSK (0.31)
SCHEMBL3788943 0.73
SCHEMBL25414924 0.72 MEN1 (0.42) MEN1KMT2A
SCHEMBL5174281 0.72 SIGMAR1 (0.40) OPRD1OPRK1STSMAPK1MEN1
SCHEMBL7345681 0.72 SMN1; SMN2 (0.40) OPRD1OPRK1STSGPR119ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3699173-A1 GEM-DISUBSTITUTED PYRROLIDINES, PIPERAZINES, AND DIAZEPANES, AND COMPOSITIONS AND METHODS OF MAKING THE SAME California Institute of Technology (US) 2020-08-26 EP disclosed