SCHEMBL2244785

SCHEMBL2244785

CCCOc1ccc(-c2ccc(C(=O)N[C@@H](CCC(=O)O)C(N)=O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.56
CA1 P00915 1/20 0.56
CA9 Q16790 1/20 0.56
MMP12 P39900 1/20 0.56
TAS1R3 Q7RTX0 2/20 0.54
TAS1R1 Q7RTX1 2/20 0.54
HPGDS O60760 1/20 0.50
PLK1 P53350 1/20 0.50
PTPN1 P18031 1/20 0.49
ADAMTS4 O75173 1/20 0.48
ADAMTS5 Q9UNA0 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48
GART P22102 3/20 0.48
FOLR2 P14207 1/20 0.48
FOLR1 P15328 1/20 0.48
SLC19A1 P41440 1/20 0.48
SLC46A1 Q96NT5 1/20 0.48
LMNA P02545 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2246121 0.95 CA12 (0.56) CA12CA1CA9MMP12TAS1R3
SCHEMBL2246912 0.91 MMP12 (0.58) CA12CA1CA9MMP12TAS1R3
SCHEMBL2244792 0.86 CA2 (0.56) CA1TAS1R3TAS1R1PLK1HRH3
SCHEMBL2251669 0.83 MMP12 (0.61) MMP12HPGDSPTPN1ADAMTS4ADAMTS5
SCHEMBL2246054 0.83 MMP12 (0.76) CA12CA1CA9MMP12HPGDS
SCHEMBL2245321 0.83 MMP12 (0.76) CA12CA1CA9MMP12HPGDS
SCHEMBL3581707 0.82 KLKB1 (0.59) MMP12ADAMTS4ADAMTS5NPC1RAB9A
SCHEMBL2249688 0.82 MMP12 (0.61) CA12CA1CA9MMP12TAS1R3
SCHEMBL2246124 0.82 CA2 (0.56) CA1TAS1R3TAS1R1HRH3GART
SCHEMBL2246545 0.81 MMP12 (0.61) CA12CA1CA9MMP12HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed