SCHEMBL2244792

SCHEMBL2244792

CCCOc1ccc(-c2ccc(C(=O)N[C@@H](CCC(N)=O)C(=O)O)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 6/20 0.56
CA1 P00915 3/20 0.56
TAS1R3 Q7RTX0 2/20 0.54
TAS1R1 Q7RTX1 2/20 0.54
PLK1 P53350 1/20 0.50
PPARG P37231 2/20 0.48
HRH3 Q9Y5N1 1/20 0.48
PPARA Q07869 1/20 0.48
GART P22102 4/20 0.48
FOLR2 P14207 1/20 0.48
FOLR1 P15328 1/20 0.48
SLC19A1 P41440 1/20 0.48
SLC46A1 Q96NT5 1/20 0.48
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
ATIC P31939 1/20 0.45
SHMT1 P34896 1/20 0.45
SHMT2 P34897 1/20 0.45
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2246124 0.95 CA2 (0.56) CA2CA1TAS1R3TAS1R1PPARG
SCHEMBL2246916 0.91 CA2 (0.58) CA2CA1TAS1R3TAS1R1PLK1
SCHEMBL2244785 0.86 CA12 (0.56) CA1TAS1R3TAS1R1PLK1PPARG
SCHEMBL2251677 0.83 GPR132 (0.55) CA2CA1
SCHEMBL2246061 0.83 CA2 (0.69) CA2CA1NPC1RAB9A
SCHEMBL2245325 0.83 CA2 (0.69) CA2CA1NPC1RAB9A
SCHEMBL2249692 0.82 CA2 (0.62) CA2CA1TAS1R3TAS1R1NPC1
SCHEMBL2246121 0.82 CA12 (0.56) CA1TAS1R3TAS1R1PPARGHRH3
SCHEMBL2246549 0.81 RXRA (0.58) CA2CA1
SCHEMBL2243990 0.81 DHFR (0.50) CA2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed