SCHEMBL22473985

SCHEMBL22473985

CCCCCCC(C)c1nc2ccccc2o1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.44
FAAH O00519 2/20 0.44
ALDH1A1 P00352 2/20 0.44
KMT2A Q03164 2/20 0.44
HSD17B10 Q99714 2/20 0.44
CES1 P23141 1/20 0.44
TP53 P04637 1/20 0.44
HSP90AA1 P07900 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
F2 P00734 1/20 0.40
LMNA P02545 1/20 0.40
MIF P14174 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HSF1 Q00613 2/20 0.39
PTGS2 P35354 1/20 0.39
HPGD P15428 1/20 0.39
CASP1 P29466 1/20 0.39
ATM Q13315 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19241750 0.98 MAPT (0.42) MAPTFAAHALDH1A1KMT2AHSD17B10
SCHEMBL27996129 0.94 MAPT (0.42) MAPTFAAHALDH1A1KMT2AHSD17B10
SCHEMBL25775949 0.88 NPC1 (0.44) MAPTFAAHALDH1A1HSD17B10CES1
SCHEMBL21118353 0.85 MAPT (0.40) MAPTALDH1A1HSD17B10TP53LMNA
SCHEMBL18626325 0.82 FAAH (0.47) FAAH
SCHEMBL13767905 0.81 RAB9A (0.47) MAPTALDH1A1TP53NPSR1LMNA
SCHEMBL9963730 0.81 RAB9A (0.47) MAPTALDH1A1TP53NPSR1LMNA
SCHEMBL15501219 0.81 HSF1 (0.39) MAPTALDH1A1HSD17B10TP53LMNA
SCHEMBL28023594 0.79 MAPT (0.42) MAPTFAAHALDH1A1KMT2AHSD17B10
SCHEMBL29780557 0.79 AAK1 (0.42) MAPTALDH1A1KMT2AHSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10787453-B2 Octahydropyrrolopyrroles their preparation and use THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2020-09-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10787453-B2 Octahydropyrrolopyrroles their preparation and use QDPR, DPYD, DHPS MAPT 1453/4885FAAH 900/4885ALDH1A1 875/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.