SCHEMBL2248654

SCHEMBL2248654

NC(=O)CC[C@H](NC(=O)c1ccc(Br)o1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.53
TAS1R1 Q7RTX1 1/20 0.53
ALDH1A1 P00352 7/20 0.51
HPGD P15428 5/20 0.51
CA2 P00918 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
CA1 P00915 2/20 0.51
POLB P06746 2/20 0.51
HTT P42858 1/20 0.51
LMNA P02545 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
NPSR1 Q6W5P4 2/20 0.48
MAPT P10636 2/20 0.47
KMT2A Q03164 2/20 0.47
C3AR1 Q16581 2/20 0.46
RAB9A P51151 3/20 0.44
NPC1 O15118 2/20 0.44
MEN1 O00255 1/20 0.44
TSHR P16473 1/20 0.44
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9380926 0.89 LMNA (0.58) TAS1R3TAS1R1ALDH1A1HPGDCA2
SCHEMBL9380922 0.89 LMNA (0.58) TAS1R3TAS1R1ALDH1A1HPGDCA2
SCHEMBL2248650 0.84 LMNA (0.56) TAS1R3TAS1R1ALDH1A1HPGDSMN1; SMN2
SCHEMBL2247803 0.82 C3AR1 (0.55) CA2CA1KMT2AC3AR1
SCHEMBL13892828 0.81 HPGD (0.72) TAS1R3TAS1R1ALDH1A1HPGDSMN1; SMN2
SCHEMBL2247341 0.78 C3AR1 (0.53) ALDH1A1CA2CA1NPSR1KMT2A
SCHEMBL2245141 0.77 C3AR1 (0.61) ALDH1A1CA2CA1NPSR1KMT2A
SCHEMBL13330083 0.77 CA2 (0.66) CA2CA1KMT2AC3AR1
SCHEMBL2244860 0.76 CA2 (0.69) CA2CA1KMT2AC3AR1
SCHEMBL2244829 0.76 S1PR4 (0.48) ALDH1A1HPGDCA2CA1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed