SCHEMBL2245141

SCHEMBL2245141

Cc1cc(C)cc(-c2ccc(C(=O)N[C@@H](CCC(N)=O)C(=O)O)o2)c1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
C3AR1 Q16581 10/20 0.61
SLC9A1 P19634 1/20 0.48
ALDH1A1 P00352 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
SUCNR1 Q9BXA5 5/20 0.47
CA2 P00918 2/20 0.45
CA1 P00915 1/20 0.45
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2247803 0.87 C3AR1 (0.55) C3AR1SUCNR1CA2CA1KMT2A
SCHEMBL2245137 0.86 C3AR1 (0.53) C3AR1SLC9A1SUCNR1CA1
SCHEMBL2243871 0.81 C3AR1 (0.75) C3AR1SLC9A1SUCNR1
SCHEMBL2246508 0.79 CA2 (0.60) C3AR1CA2CA1KMT2A
SCHEMBL2247341 0.78 C3AR1 (0.53) C3AR1ALDH1A1NPSR1SUCNR1CA2
SCHEMBL2248654 0.77 TAS1R3 (0.53) C3AR1ALDH1A1NPSR1CA2CA1
SCHEMBL3581142 0.77 MMP2 (0.47) C3AR1ALDH1A1CA2CA1
SCHEMBL2244829 0.76 S1PR4 (0.48) C3AR1ALDH1A1NPSR1CA2CA1
SCHEMBL23091227 0.76 CYP1A2 (0.59) C3AR1SLC9A1ALDH1A1SUCNR1KMT2A
SCHEMBL26263216 0.75 C3AR1 (0.67) C3AR1SLC9A1SUCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed