SCHEMBL22497768

SCHEMBL22497768

CC1(C)OB(c2cc(F)c3c(c2)CCC3=O)OC1(C)C

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.39
LPL P06858 4/20 0.37
LIPG Q9Y5X9 4/20 0.37
BACE1 P56817 2/20 0.32
P2RX7 Q99572 1/20 0.32
CA1 P00915 3/20 0.31
CA2 P00918 3/20 0.31
CA9 Q16790 3/20 0.31
CA12 O43570 1/20 0.31
CA3 P07451 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31
CA5A P35218 1/20 0.31
CA7 P43166 1/20 0.31
CA14 Q9ULX7 1/20 0.31
CA5B Q9Y2D0 1/20 0.31
MAPK1 P28482 1/20 0.30
JAK2 O60674 1/20 0.30
BTK Q06187 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27157750 0.81 ROCK1 (0.36) ROCK1LPLLIPGJAK2
SCHEMBL6127173 0.81 LPL (0.41) ROCK1LPLLIPGP2RX7CA1
SCHEMBL21493489 0.77 KIF11 (0.39) ROCK1LPLLIPGBACE1P2RX7
SCHEMBL1477653 0.77 ROCK1 (0.37) ROCK1LPLLIPGJAK2
SCHEMBL28347176 0.76 ROCK1 (0.42) ROCK1LPLLIPG
SCHEMBL14778585 0.75 ROCK1 (0.38) ROCK1LPLLIPGBACE1JAK2
SCHEMBL17233424 0.74 ROCK1 (0.34) ROCK1LPLLIPG
SCHEMBL25118557 0.73 LIPG (0.43) ROCK1LPLLIPGBACE1P2RX7
SCHEMBL15726606 0.73 LPL (0.36) LPLLIPGBACE1P2RX7CA1
SCHEMBL483144 0.73 CASP1 (0.45) ROCK1LPLLIPGBACE1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113544129-A Tricyclic compound preparation method and application thereof in medicine field 上海华汇拓医药科技有限公司 2021-10-22 CN disclosed
WO-2020200284-A1 PREPARATION METHOD FOR TRICYCLIC COMPOUND AND USE OF SAME IN FIELD OF MEDICINE 上海华汇拓医药科技有限公司 2020-10-08 WO disclosed