SCHEMBL22556882

SCHEMBL22556882

NC(=O)C(O)c1ccc(N)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.41
ADRA2B P18089 2/20 0.41
ADRA2C P18825 2/20 0.41
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA13 Q8N1Q1 1/20 0.38
CA14 Q9ULX7 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.34
NNMT P40261 1/20 0.34
PTGS1 P23219 2/20 0.34
APLNR P35414 1/20 0.33
MKNK1 Q9BUB5 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
GABRP O00591 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19717001 0.78 APLNR (0.53) APLNRGABRA5
SCHEMBL19716497 0.78 ADRA2A (0.43) ADRA2AADRA2BADRA2CSMN1; SMN2APLNR
SCHEMBL29658558 0.78 ADRA2A (0.43) ADRA2AADRA2BADRA2CSMN1; SMN2APLNR
SCHEMBL9649808 0.78 ADRB2 (0.37) ADRA2AADRA2BADRA2CCA12CA1
SCHEMBL20644139 0.77 ADRA2A (0.41) ADRA2AADRA2BADRA2CCA12CA1
SCHEMBL2068072 0.75 HTT (0.43) ADRA2AADRA2BADRA2CSMN1; SMN2L3MBTL1
SCHEMBL22556951 0.75 ADRA2A (0.39) ADRA2AADRA2BADRA2CCA12CA1
SCHEMBL15466329 0.74 PANK3 (0.40) LMNAL3MBTL1KDM4EMEN1KMT2A
SCHEMBL19716796 0.74 CACNA1I (0.44) CA1CA2NNMTKDM4E
SCHEMBL22557408 0.74 ALDH1A1 (0.34) ADRA2AADRA2BADRA2CCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3956322-A1 JAK1 SELECTIVE KINASE INHIBITOR DIZAL (JIANGSU) PHARMACEUTICAL CO., LTD. (CN) 2022-02-23 EP disclosed
WO-2020211839-A1 JAK1 SELECTIVE KINASE INHIBITOR DIZAL (JIANGSU) PHARMACEUTICAL CO., LTD. (CN) 2020-10-22 WO disclosed