SCHEMBL22562946

SCHEMBL22562946

Cc1ccc(Nc2ccc(C(=N)C(C)C)c(N)c2)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K2 P36507 1/20 0.39
MAP2K1 Q02750 1/20 0.39
DHODH Q02127 9/20 0.36
GAA P10253 4/20 0.36
KDM4E B2RXH2 3/20 0.36
MAPT P10636 3/20 0.36
GFER P55789 2/20 0.36
NPC1 O15118 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 2/20 0.33
MAPK13 O15264 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK11 Q15759 1/20 0.33
MAPK14 Q16539 1/20 0.33
CSF1R P07333 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562967 0.86 NUDT1 (0.37) MAP2K1GAAKDM4EMAPTGFER
SCHEMBL22563002 0.86 MAP2K2 (0.41) MAP2K2MAP2K1DHODHGAAKDM4E
SCHEMBL22563054 0.85 MAPK14 (0.40) GAAKDM4EMAPTSMN1; SMN2HSD17B10
SCHEMBL22562957 0.83 MAP2K1 (0.41) MAP2K1GAAKDM4EMEN1KMT2A
SCHEMBL22563085 0.79 PYGL (0.41) GAATDP1MAPK13MAPK12MAPK11
SCHEMBL22563010 0.77 HDAC6 (0.37) MAPK13MAPK12MAPK11MAPK14HDAC1
SCHEMBL22563088 0.74 MAPK14 (0.44) GAAMAPTKMT2ATDP1MAPK13
SCHEMBL22562974 0.74 TAS2R14 (0.42) GAAKDM4EMAPTGFERSMN1; SMN2
SCHEMBL18590739 0.72 SOS1 (0.46) MAP2K2MAP2K1DHODHGAAKDM4E
SCHEMBL22563163 0.72 HDAC1 (0.40) MAP2K1GAAKDM4EMAPTGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed