SCHEMBL22563088

SCHEMBL22563088

CC(C)C(=N)c1ccc(Nc2ccccc2Cl)cc1N

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 12/20 0.44
MAPK13 O15264 8/20 0.44
MAPK12 P53778 8/20 0.44
MAPK11 Q15759 8/20 0.44
GAA P10253 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
ALDH1A1 P00352 1/20 0.37
ALOX15 P16050 1/20 0.37
HTT P42858 1/20 0.37
MAPK8 P45983 2/20 0.36
MAPK10 P53779 2/20 0.36
KMT2A Q03164 1/20 0.36
ACVRL1 P37023 1/20 0.36
AURKA O14965 2/20 0.35
AURKB Q96GD4 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562988 0.85 MAPK14 (0.47) MAPK14MAPK13MAPK12MAPK11GAA
SCHEMBL22563054 0.84 MAPK14 (0.40) MAPK14MAPK13MAPK12MAPK11GAA
SCHEMBL22563085 0.84 PYGL (0.41) MAPK14MAPK13MAPK12MAPK11GAA
SCHEMBL22562974 0.81 TAS2R14 (0.42) MAPK14MAPK13MAPK12MAPK11GAA
SCHEMBL22562967 0.79 NUDT1 (0.37) GAAHTTKMT2AMAPT
SCHEMBL22562946 0.74 MAP2K2 (0.39) MAPK14MAPK13MAPK12MAPK11GAA
SCHEMBL22563010 0.71 HDAC6 (0.37) MAPK14MAPK13MAPK12MAPK11
SCHEMBL22562957 0.71 MAP2K1 (0.41) GAAALDH1A1KMT2A
SCHEMBL22563179 0.69 HDAC1 (0.44) MAPK14MAPK13MAPK12MAPK11GAA
SCHEMBL22563042 0.68 PYGL (0.44) MAPK14MAPK13MAPK12MAPK11GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed