SCHEMBL22562967

SCHEMBL22562967

CC(C)C(=N)c1ccc(Nc2ccc(Cl)cc2F)cc1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 3/20 0.37
MAP2K1 Q02750 2/20 0.37
CNR2 P34972 1/20 0.36
KMT2A Q03164 6/20 0.36
MEN1 O00255 4/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
GFER P55789 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ABL1 P00519 1/20 0.36
HDAC1 Q13547 1/20 0.35
RAB9A P51151 1/20 0.34
CSF1R P07333 1/20 0.34
MAPT P10636 2/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562946 0.86 MAP2K2 (0.39) MAP2K1KMT2AMEN1KDM4EGAA
SCHEMBL22563163 0.86 HDAC1 (0.40) NUDT1MAP2K1CNR2KMT2AMEN1
SCHEMBL22563054 0.84 MAPK14 (0.40) KDM4EGAAHSD17B10HDAC1RAB9A
SCHEMBL22563085 0.83 PYGL (0.41) CNR2GAAHDAC1CSF1RHTT
SCHEMBL22562957 0.82 MAP2K1 (0.41) MAP2K1KMT2AMEN1KDM4EGAA
SCHEMBL22563088 0.79 MAPK14 (0.44) KMT2AGAAMAPTHTT
SCHEMBL22563010 0.73 HDAC6 (0.37) HDAC1LMNA
SCHEMBL22562974 0.73 TAS2R14 (0.42) KMT2AMEN1KDM4EGAAGFER
SCHEMBL22563002 0.72 MAP2K2 (0.41) MAP2K1KMT2AMEN1KDM4EGAA
SCHEMBL22562958 0.71 JAK1 (0.37) KMT2AMEN1KDM4EHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed