SCHEMBL22562973

SCHEMBL22562973

CCCCC(CCC)c1ccc(C(=O)NC(NC)c2ccc(Nc3ccc(C)cc3)cc2N)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
GFER P55789 1/20 0.36
SCN5A Q14524 1/20 0.35
SCN2A Q99250 1/20 0.35
CA2 P00918 1/20 0.35
ERAP2 Q6P179 3/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
RECQL P46063 1/20 0.33
PLAU P00749 1/20 0.33
HPN P05981 1/20 0.33
HTT P42858 1/20 0.32
LNPEP Q9UIQ6 2/20 0.32
TAS1R3 Q7RTX0 4/20 0.32
TAS1R1 Q7RTX1 4/20 0.32
UTS2R Q9UKP6 3/20 0.32
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22563056 0.67 HDAC1 (0.41) MAPTKDM4ENPC1MEN1KMT2A
SCHEMBL3289894 0.66 HRH3 (0.45) CA2HTT
SCHEMBL22563013 0.66 MAPK14 (0.41) KDM4ENPC1GAAGFERMEN1
SCHEMBL28533240 0.64 BDKRB2 (0.49) TAS1R3TAS1R1
SCHEMBL22563037 0.63 RARB (0.47) MAPTMEN1KMT2A
SCHEMBL8759863 0.62 NR1I2 (0.47) MAPTSMN1; SMN2MEN1KMT2A
SCHEMBL21078080 0.62 TAS1R3 (0.58) SMN1; SMN2GAASCN5ASCN2ACA2
SCHEMBL28863365 0.61 MEN1 (0.53) MAPTSMN1; SMN2NPC1GAASCN5A
SCHEMBL28836790 0.61 HSD17B10 (0.46) SMN1; SMN2NPC1CA2MEN1KMT2A
SCHEMBL21711047 0.61 TAS1R3 (0.73) SMN1; SMN2HTTTAS1R3TAS1R1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed