SCHEMBL22562963

SCHEMBL22562963

CCCCCC(CCC)c1ccc(C(=O)N/C(=C(/C)CC)c2ccc(Nc3ccccc3C)cc2N)cc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 10/20 0.39
MAPK13 O15264 6/20 0.39
MAPK12 P53778 6/20 0.39
MAPK11 Q15759 6/20 0.39
HDAC1 Q13547 5/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC2 Q92769 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
EPHX1 P07099 1/20 0.32
PLK1 P53350 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22563056 0.82 HDAC1 (0.41) HDAC1NPC1RAB9AMEN1KMT2A
SCHEMBL22562998 0.80 MAPK14 (0.33) MAPK14MAPK13MAPK12MAPK11HDAC1
SCHEMBL22563055 0.74 TBXA2R (0.38) HDAC1MEN1KMT2AALDH1A1MAPT
SCHEMBL22563033 0.72 MAPK14 (0.47) MAPK14MAPK13MAPK12MAPK11HDAC1
SCHEMBL22563017 0.72 HDAC1 (0.37) MAPK14MAPK13MAPK12MAPK11HDAC1
SCHEMBL22563043 0.68 ALDH1A1 (0.35) HDAC1NPC1RAB9AMEN1KMT2A
SCHEMBL9799041 0.66 MAPK14 (0.59) MAPK14MAPK13MAPK12MAPK11NPC1
SCHEMBL22563034 0.66 HDAC1 (0.37) HDAC1HDAC3HDAC2ALDH1A1
SCHEMBL12172229 0.63 NR1I2 (0.47) KMT2AL3MBTL1
SCHEMBL27718637 0.63 MAPK13 (0.59) MAPK14MAPK13MAPK12MAPK11NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed