SCHEMBL22563055

SCHEMBL22563055

CCCCC(CCC)c1ccc(C(=O)N/C(=C(/C)CC)c2ccc(Nc3ccc(C#N)cc3C)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 7/20 0.38
HDAC1 Q13547 1/20 0.34
MAP2K1 Q02750 2/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
NAMPT P43490 2/20 0.32
ALDH1A1 P00352 1/20 0.32
PKM P14618 1/20 0.32
CTSG P08311 1/20 0.32
EPHX2 P34913 1/20 0.31
SCN5A Q14524 1/20 0.31
SCN2A Q99250 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562963 0.74 MAPK14 (0.39) HDAC1KMT2AMEN1ALDH1A1MAPT
SCHEMBL22563056 0.68 HDAC1 (0.41) HDAC1KMT2AMEN1MAPT
SCHEMBL22563043 0.66 ALDH1A1 (0.35) HDAC1KMT2AMEN1NAMPTALDH1A1
SCHEMBL21783907 0.63 TSHR (0.46) ALDH1A1
SCHEMBL28533240 0.61 BDKRB2 (0.49) ALDH1A1
SCHEMBL18432620 0.61 CYP2A6 (0.48) ALDH1A1MAPT
SCHEMBL8131540 0.60 TSHR (0.50) ALDH1A1
SCHEMBL22563037 0.60 RARB (0.47) KMT2AMEN1ALDH1A1MAPT
SCHEMBL20303234 0.60 KDM4E (0.54) KMT2AMEN1ALDH1A1MAPT
SCHEMBL19232073 0.60 TSHR (0.49) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed