SCHEMBL2260449

SCHEMBL2260449

CC(C)NC(=O)c1cc(O)cc(-c2ccc3c(c2)OCO3)c1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
GABRA1 P14867 1/20 0.50
GABRB2 P47870 1/20 0.50
TAS1R3 Q7RTX0 7/20 0.47
TAS1R1 Q7RTX1 7/20 0.47
ADORA3 P0DMS8 3/20 0.46
ADORA1 P30542 2/20 0.46
GAA P10253 1/20 0.45
KMT2A Q03164 1/20 0.45
HPGD P15428 1/20 0.44
CTSA P10619 1/20 0.44
ADORA2A P29274 1/20 0.44
ERN1 O75460 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2260517 0.86 KDM4E (0.52) GABRA1GABRB2TAS1R3TAS1R1GAA
SCHEMBL200964 0.84 GABRA1 (0.54) NPC1RAB9AGABRA1GABRB2ADORA3
SCHEMBL2262131 0.81 RAB9A (0.60) NPC1RAB9AGAAKMT2AHPGD
SCHEMBL2261168 0.81 NPC1 (0.62) NPC1RAB9AKMT2AHPGDERN1
SCHEMBL2260303 0.81 NPC1 (0.65) NPC1RAB9AADORA3ADORA1KMT2A
SCHEMBL2261442 0.80 MCHR1 (0.59) NPC1RAB9AGABRA1GABRB2ADORA3
SCHEMBL2260433 0.80 NPC1 (0.67) NPC1RAB9AKMT2AHPGDERN1
SCHEMBL2262389 0.80 AKR1C4 (0.48) NPC1RAB9AGABRA1GABRB2ADORA3
SCHEMBL11142926 0.80 TAS1R3 (0.67) NPC1RAB9ATAS1R3TAS1R1KMT2A
SCHEMBL2261354 0.79 NPC1 (0.66) NPC1RAB9AKMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989454-B2 Leukotriene B4 inhibitors HOFFMANN-LA ROCHE INC. (US) 2011-08-02 US disclosed
US-7989454-B2 Leukotriene B4 inhibitors HOFFMANN-LA ROCHE INC. (US) 2011-08-02 US disclosed
US-7989454-B2 Leukotriene B4 inhibitors HOFFMANN-LA ROCHE INC. (US) 2011-08-02 US disclosed
US-20090253684-A1 LEUKOTRIENE B4 INHIBITORS DOMINIQUE ROMYR 2009-10-08 US disclosed
US-20090253684-A1 LEUKOTRIENE B4 INHIBITORS DOMINIQUE ROMYR 2009-10-08 US disclosed
US-20090253684-A1 LEUKOTRIENE B4 INHIBITORS DOMINIQUE ROMYR 2009-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090253684-A1 LEUKOTRIENE B4 INHIBITORS LTB4R2, LTB4R, LTC4S NPC1 689/4885RAB9A 3108/4885GABRA1 1497/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.