SCHEMBL22604799

SCHEMBL22604799

C=CC(=O)Nc1cccc(Sc2nc(Nc3ccc(C)cc3)ncc2Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BTK Q06187 8/20 0.62
EGFR P00533 10/20 0.61
JAK3 P52333 2/20 0.56
ITK Q08881 3/20 0.54
MAP3K7 O43318 1/20 0.53
MAP2K1 Q02750 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22604617 0.92 EGFR (0.59) BTKEGFRJAK3ITKMAP3K7
SCHEMBL93523 0.85 MAP3K7 (0.74) BTKEGFRJAK3MAP3K7MAP2K1
SCHEMBL29352639 0.85 MAP3K7 (0.74) BTKEGFRJAK3MAP3K7MAP2K1
SCHEMBL30854787 0.85 MAP3K7 (0.74) BTKEGFRJAK3MAP3K7MAP2K1
SCHEMBL13165510 0.85 BTK (0.69) BTKEGFRJAK3ITK
SCHEMBL28080977 0.78 BTK (0.88) BTKEGFRJAK3ITK
SCHEMBL27831797 0.76 EGFR (0.84) BTKEGFRJAK3ITK
SCHEMBL28059266 0.76 EGFR (0.77) BTKEGFRITK
SCHEMBL10127876 0.75 JAK3 (0.80) BTKEGFRJAK3ITK
SCHEMBL13169901 0.75 EGFR (0.58) BTKEGFRJAK3ITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020219963-A1 METHODS AND COMPOSITIONS FOR TREATING CHRONIC INFLAMMATORY INJURY, METAPLASIA, DYSPLASIA AND CANCERS OF EPITHELIAL TISSUES UNIVERSITY OF HOUSTON SYSTEM (US) 2020-10-29 WO disclosed