SCHEMBL22607366

SCHEMBL22607366

Cc1ccc(C(C)C)cc1N(C)CCN(C)C

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.44
TRPA1 O75762 1/20 0.43
PTGS1 P23219 1/20 0.43
CACNA1C Q13936 1/20 0.43
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
ACHE P22303 4/20 0.38
BCHE P06276 3/20 0.38
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
HTT P42858 1/20 0.33
UTS2R Q9UKP6 1/20 0.33
C5AR1 P21730 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18999634 0.83 HTR1D (0.40) LMNATRPA1PTGS1CACNA1CHTR1D
SCHEMBL21969437 0.80 HTR1D (0.41) LMNAHTR1DHTR1BACHEBCHE
SCHEMBL19007315 0.78 HTT (0.39) LMNATRPA1SMN1; SMN2KDM4EALDH1A1
SCHEMBL23983215 0.78 ALDH1A1 (0.44) LMNAHTR1DHTR1BHPGDSMN1; SMN2
SCHEMBL14228579 0.77 LMNA (0.54) LMNATRPA1PTGS1CACNA1CACHE
SCHEMBL13130519 0.76 HTR1D (0.38) LMNAHTR1DHTR1BHPGDSMN1; SMN2
SCHEMBL23520055 0.74 LMNA (0.50) LMNATRPA1PTGS1CACNA1CACHE
SCHEMBL8148875 0.73 TRPA1 (0.36) LMNATRPA1PTGS1CACNA1CACHE
SCHEMBL26514879 0.73 LMNA (0.48) LMNATRPA1PTGS1CACNA1CACHE
SCHEMBL12648604 0.72 HPGD (0.42) HTR1DHTR1BHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3122353-B1 SUBSTITUTED INDOLE MCL-1 INHIBITORS UNIV VANDERBILT (US) 2020-10-28 EP disclosed