SCHEMBL22650385

SCHEMBL22650385

CC(C)(C)OC(=O)N1CCN(c2ccc(N)c(F)c2F)C(=O)C1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.44
MAPT P10636 2/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE7A Q13946 1/20 0.41
SMARCA2 P51531 1/20 0.40
SMARCA4 P51532 1/20 0.40
PBRM1 Q86U86 1/20 0.40
ESR2 Q92731 1/20 0.39
P2RX7 Q99572 7/20 0.39
ADORA1 P30542 1/20 0.39
MAPK1 P28482 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HDAC2 Q92769 4/20 0.38
HDAC1 Q13547 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1662799 0.86 NR1H2 (0.41) NR1H2MAPTALDH1A1LMNAPDE4B
SCHEMBL31487442 0.84 MAPT (0.51) NR1H2MAPTALDH1A1LMNASMARCA2
SCHEMBL21245582 0.84 MAPT (0.51) NR1H2MAPTALDH1A1LMNASMARCA2
SCHEMBL22650493 0.82 NR1H2 (0.54) NR1H2PDE4BPDE7AESR2P2RX7
SCHEMBL29507776 0.82 NR1H2 (0.54) NR1H2PDE4BPDE7AESR2P2RX7
SCHEMBL4537183 0.81 P2RX7 (0.55) P2RX7
SCHEMBL1583488 0.81 MEN1 (0.51) NR1H2MAPTP2RX7MAPK1KDM4E
SCHEMBL30734152 0.81 MEN1 (0.51) NR1H2MAPTP2RX7MAPK1KDM4E
SCHEMBL22650491 0.80 NR1H2 (0.46) NR1H2MAPTALDH1A1LMNASMARCA2
SCHEMBL1662960 0.80 P2RX7 (0.44) NR1H2MAPTLMNAPDE4BPDE7A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed