SCHEMBL1662799

SCHEMBL1662799

COc1ccc(N2CCN(C(=O)OC(C)(C)C)CC2=O)c(F)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.41
P2RX7 Q99572 2/20 0.41
RBP4 P02753 1/20 0.40
PDE4B Q07343 5/20 0.40
PDE7A Q13946 1/20 0.40
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
PDE4A P27815 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
ALDH1A1 P00352 2/20 0.38
ESR2 Q92731 1/20 0.38
STS P08842 1/20 0.38
ADORA1 P30542 1/20 0.38
F13A1 P00488 1/20 0.38
TGM2 P21980 1/20 0.38
TGM1 P22735 1/20 0.38
SMPD3 Q9NY59 1/20 0.38
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650385 0.86 NR1H2 (0.44) NR1H2P2RX7PDE4BPDE7AMAPT
SCHEMBL1663317 0.82 NR1H2 (0.40) NR1H2P2RX7RBP4PDE4BPDE7A
SCHEMBL1662800 0.81 PTGDR2 (0.44) P2RX7RBP4MAPTALDH1A1LMNA
SCHEMBL1584703 0.81 CPS1 (0.46) NR1H2P2RX7MAPTKDM4EALDH1A1
SCHEMBL1663275 0.81 GALR2 (0.43) NR1H2PDE4BMAPTKDM4EPDE4A
SCHEMBL4537183 0.79 P2RX7 (0.55) P2RX7MKNK1
SCHEMBL1583488 0.79 MEN1 (0.51) NR1H2P2RX7MAPTKDM4EMAPK1
SCHEMBL30734152 0.79 MEN1 (0.51) NR1H2P2RX7MAPTKDM4EMAPK1
SCHEMBL1662960 0.78 P2RX7 (0.44) NR1H2P2RX7PDE4BPDE7AMAPT
SCHEMBL22650493 0.78 NR1H2 (0.54) NR1H2P2RX7PDE4BPDE7AESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050284-A1 PYRAZOLYLPYRIDINE ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2011-04-28 WO disclosed