SCHEMBL22650455

SCHEMBL22650455

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5CCC(C)(N)CC5=O)cc4Cl)n3)cc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 7/20 0.35
PIK3CA P42336 4/20 0.35
PIK3CB P42338 4/20 0.35
CDK1 P06493 3/20 0.34
CDK4 P11802 3/20 0.34
CCNB1 P14635 3/20 0.34
CCND1 P24385 3/20 0.34
CDK6 Q00534 1/20 0.34
MAPK3 P27361 4/20 0.33
MAPK1 P28482 4/20 0.33
BTK Q06187 1/20 0.33
MAPK8 P45983 2/20 0.32
CAMKK2 Q96RR4 2/20 0.32
TTK P33981 1/20 0.32
MAP3K14 Q99558 1/20 0.32
JAK2 O60674 1/20 0.32
ALK Q9UM73 1/20 0.32
ABL1 P00519 1/20 0.31
BCR P11274 1/20 0.31
CCNA2 P20248 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650715 0.92 CDK6 (0.35) PIK3CGPIK3CAPIK3CBCDK1CDK4
SCHEMBL22650766 0.89 JAK2 (0.39) CDK1CDK4CCNB1CCND1CDK6
SCHEMBL22650755 0.89 CDK4 (0.42) CDK1CDK4CCNB1CCND1CDK6
SCHEMBL22650705 0.77 CDK6 (0.39) CDK1CDK4CCNB1CCND1CDK6
SCHEMBL22650937 0.77 CDK4 (0.40) CDK1CDK4CCNB1CCND1CDK6
SCHEMBL22650524 0.76 CDK6 (0.38) CDK1CDK4CCNB1CCND1CDK6
SCHEMBL22650922 0.76 F10 (0.38) MAPK8MAP3K14JAK2
SCHEMBL22650453 0.75 CDK4 (0.42) CDK1CDK4CCNB1CCND1CDK6
SCHEMBL22650846 0.75 CDK4 (0.42) CDK1CDK4CCNB1CCND1CDK6
SCHEMBL29491175 0.75 CDK4 (0.49) CDK1CDK4CCNB1CCND1CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed