SCHEMBL22650467

SCHEMBL22650467

O=C1COCCN1c1ccc(Nc2ncc(F)c(-c3ccn4ncc(C5CCCC5)c4c3)n2)nc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 15/20 0.49
CCND1 P24385 11/20 0.49
CDK6 Q00534 10/20 0.44
CCND3 P30281 5/20 0.44
CDK1 P06493 2/20 0.44
CCNA2 P20248 2/20 0.44
TYK2 P29597 2/20 0.44
JAK2 O60674 1/20 0.44
JAK1 P23458 1/20 0.44
JAK3 P52333 1/20 0.44
PIM1 P11309 1/20 0.42
CCNB1 P14635 1/20 0.42
CDK2 P24941 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650471 0.95 CDK4 (0.46) CDK4CCND1CDK6CCND3CDK1
SCHEMBL22650591 0.86 CDK6 (0.48) CDK4CCND1CDK6CCND3CDK1
SCHEMBL22650928 0.84 CDK6 (0.50) CDK4CCND1CDK6CCND3CDK1
SCHEMBL22650468 0.83 CDK6 (0.41) CDK4CCND1CDK6CCND3CDK1
SCHEMBL22650401 0.76 NTRK1 (0.46) CDK4CDK6CCNA2JAK2JAK1
SCHEMBL22650487 0.75 CDK4 (0.42) CDK4CDK6CCNA2TYK2JAK2
SCHEMBL22650845 0.74 CDK6 (0.48) CDK4CCND1CDK6CCND3CDK1
SCHEMBL29491166 0.73 CDK6 (0.55) CDK4CCND1CDK6CCND3CDK1
SCHEMBL22650475 0.73 CDK6 (0.58) CDK4CCND1CDK6CCND3CDK1
SCHEMBL22650846 0.73 CDK4 (0.42) CDK4CCND1CDK6CCND3CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed