SCHEMBL22650471

SCHEMBL22650471

O=C1COCCN1c1ccc(Nc2ncc(F)c(-c3ccn4ncc(C5CCOCC5)c4c3)n2)nc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 13/20 0.46
CCND1 P24385 8/20 0.46
CDK6 Q00534 15/20 0.44
TYK2 P29597 2/20 0.44
JAK2 O60674 1/20 0.44
JAK1 P23458 1/20 0.44
JAK3 P52333 1/20 0.44
PIM1 P11309 2/20 0.44
CCND3 P30281 5/20 0.43
CCNA2 P20248 3/20 0.43
CDK1 P06493 2/20 0.43
CDK2 P24941 2/20 0.42
PIK3CD O00329 1/20 0.42
CCNK O75909 1/20 0.42
CSF1R P07333 1/20 0.42
CDK9 P50750 1/20 0.42
CCNB1 P14635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650467 0.95 CDK4 (0.49) CDK4CCND1CDK6TYK2JAK2
SCHEMBL22650591 0.86 CDK6 (0.48) CDK4CCND1CDK6TYK2JAK2
SCHEMBL22650928 0.84 CDK6 (0.50) CDK4CCND1CDK6PIM1CCND3
SCHEMBL22650468 0.83 CDK6 (0.41) CDK4CCND1CDK6TYK2JAK2
SCHEMBL22650401 0.76 NTRK1 (0.46) CDK4CDK6JAK2JAK1JAK3
SCHEMBL22650487 0.75 CDK4 (0.42) CDK4CDK6TYK2JAK2JAK1
SCHEMBL22650475 0.75 CDK6 (0.58) CDK4CCND1CDK6PIM1CCND3
SCHEMBL22650845 0.74 CDK6 (0.48) CDK4CCND1CDK6CCND3CCNA2
SCHEMBL22650945 0.73 CDK6 (0.60) CDK4CCND1CDK6PIM1CCND3
SCHEMBL22650846 0.73 CDK4 (0.42) CDK4CCND1CDK6TYK2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed