SCHEMBL22650468

SCHEMBL22650468

O=C1COCCN1c1ccc(Nc2ncc(F)c(-c3ccn4ncc(C5=CCOCC5)c4c3)n2)nc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 18/20 0.41
CDK4 P11802 13/20 0.41
CCND3 P30281 9/20 0.41
CCND1 P24385 8/20 0.41
CCNA2 P20248 7/20 0.41
CDK2 P24941 5/20 0.41
CDK9 P50750 5/20 0.41
CCNT1 O60563 4/20 0.41
CDK7 P50613 3/20 0.41
CCNH P51946 3/20 0.41
MNAT1 P51948 3/20 0.41
TYK2 P29597 2/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
JAK3 P52333 1/20 0.41
PIM1 P11309 2/20 0.40
CDK1 P06493 2/20 0.39
PIK3CD O00329 1/20 0.39
CCNK O75909 1/20 0.39
CSF1R P07333 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650591 0.83 CDK6 (0.48) CDK6CDK4CCND3CCND1CCNA2
SCHEMBL22650471 0.83 CDK4 (0.46) CDK6CDK4CCND3CCND1CCNA2
SCHEMBL22650467 0.83 CDK4 (0.49) CDK6CDK4CCND3CCND1CCNA2
SCHEMBL22650698 0.75 MAPK14 (0.35) CDK2PIK3CD
SCHEMBL22650401 0.74 NTRK1 (0.46) CDK6CDK4CCNA2CDK2JAK2
SCHEMBL22650487 0.73 CDK4 (0.42) CDK6CDK4CCNA2CDK2CDK9
SCHEMBL22650928 0.72 CDK6 (0.50) CDK6CDK4CCND3CCND1CCNA2
SCHEMBL22650601 0.72 CDK6 (0.48) CDK6CDK4CCND3CCND1CCNA2
SCHEMBL22650486 0.72 CDK6 (0.54) CDK6CDK4CCND3CCND1CCNA2
SCHEMBL29491147 0.72 CDK6 (0.54) CDK6CDK4CCND3CCND1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed