SCHEMBL22650618

SCHEMBL22650618

CC(C)n1cnc2c(F)nc(-c3ccnc(Nc4ccc(N5CCC(C)(N)CC5=O)cc4Cl)n3)cc21

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TTK P33981 1/20 0.33
EGFR P00533 1/20 0.32
CDK4 P11802 2/20 0.32
CCND1 P24385 2/20 0.32
CCND3 P30281 2/20 0.32
CDK6 Q00534 2/20 0.32
PIK3CG P48736 4/20 0.31
PIK3CA P42336 3/20 0.31
PIK3CB P42338 3/20 0.31
MAPK3 P27361 1/20 0.30
MAPK1 P28482 1/20 0.30
IDH1 O75874 1/20 0.30
ALK Q9UM73 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650624 0.93 EGFR (0.34) EGFRCCND3CDK6
SCHEMBL22650777 0.89 ACVR1 (0.35) TTKEGFRCDK4CDK6MAPK1
SCHEMBL22650576 0.88 CDK6 (0.38) CDK4CCND1CCND3CDK6
SCHEMBL22650513 0.79 CDK4 (0.36) CDK4CCND1CCND3CDK6
SCHEMBL22650455 0.76 PIK3CG (0.35) TTKCDK4CCND1CDK6PIK3CG
SCHEMBL22650541 0.75 EGFR (0.36) EGFRCDK4CCND1ALK
SCHEMBL22650532 0.75 EGFR (0.36) EGFRCDK4CCND1CCND3CDK6
SCHEMBL22650875 0.74 TYK2 (0.44) CDK4CCND1CCND3CDK6
SCHEMBL22650579 0.74 CDK4 (0.48) CDK4CCND1CCND3CDK6
SCHEMBL22650778 0.73 CDK4 (0.42) CDK4CCND1CCND3CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed