SCHEMBL22650818

SCHEMBL22650818

Nc1ccc(N2CCC(N3CCOCC3)CC2=O)cn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.37
MTOR P42345 8/20 0.37
PIK3R1 P27986 6/20 0.37
AKT1 P31749 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
RICTOR Q6R327 5/20 0.36
RPTOR Q8N122 5/20 0.36
MAPKAP1 Q9BPZ7 5/20 0.36
MLST8 Q9BVC4 5/20 0.36
ACVR1 Q04771 1/20 0.36
TSHR P16473 1/20 0.35
MAP4K4 O95819 1/20 0.35
HRH3 Q9Y5N1 3/20 0.35
L3MBTL3 Q96JM7 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35
HRH1 P35367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650819 0.88 HRH3 (0.39) HRH3L3MBTL3L3MBTL1HRH1
SCHEMBL22650822 0.82 CHRNB2 (0.37) HRH3HRH1
SCHEMBL22650820 0.81 CHRNB2 (0.34) HRH3L3MBTL3ALOX5APFEN1HRH1
SCHEMBL29437377 0.80 L3MBTL3 (0.50) PIK3CAMTORPIK3R1AKT1ACVR1
SCHEMBL2723240 0.80 L3MBTL3 (0.50) PIK3CAMTORPIK3R1AKT1ACVR1
SCHEMBL12280261 0.77 PIK3CA (0.43) PIK3CAMTORPIK3R1AKT1TDP1
SCHEMBL22650564 0.77 HRH3 (0.44) TSHRHRH3L3MBTL1ALDH1A1MAPK1
SCHEMBL22650730 0.76 ALOX5AP (0.40) PIK3CAMTORHRH3ALDH1A1ALOX5AP
SCHEMBL29462406 0.76 F10 (0.49) PIK3CAMTORPIK3R1
SCHEMBL2343226 0.76 F10 (0.49) PIK3CAMTORPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed