SCHEMBL22650822

SCHEMBL22650822

Nc1ccc(N2CCC(N3CC(F)C3)CC2=O)cn1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
HRH3 Q9Y5N1 6/20 0.34
GCKR Q14397 1/20 0.33
HRH1 P35367 1/20 0.33
MGLL Q99685 1/20 0.33
AKR1C3 P42330 1/20 0.32
DPP4 P27487 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650819 0.86 HRH3 (0.39) CHRNB2CHRNA4HRH3HRH1MGLL
SCHEMBL22650820 0.84 CHRNB2 (0.34) CHRNB2CHRNA4HRH3HRH1MGLL
SCHEMBL22650818 0.82 PIK3CA (0.37) HRH3HRH1
SCHEMBL22650730 0.76 ALOX5AP (0.40) CHRNB2CHRNA4HRH3GCKRAKR1C3
SCHEMBL22650564 0.74 HRH3 (0.44) HRH3
SCHEMBL22650368 0.73 ALOX5AP (0.37) CHRNB2CHRNA4GCKRAKR1C3
SCHEMBL29462389 0.73 ALOX5AP (0.37) CHRNB2CHRNA4GCKRAKR1C3
SCHEMBL22650561 0.72 TP53 (0.31) CHRNB2CHRNA4GCKRAKR1C3
SCHEMBL12425528 0.71 CHRNB2 (0.43) CHRNB2CHRNA4
SCHEMBL12425903 0.71 CHRNB2 (0.43) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed