SCHEMBL22702191

SCHEMBL22702191

CC(C)/C(N)=C/NCc1ccccn1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
SMN1; SMN2 Q16637 2/20 0.45
CYP1A2 P05177 3/20 0.44
POLB P06746 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPT P10636 1/20 0.44
TSHR P16473 1/20 0.44
MAOA P21397 3/20 0.42
MAOB P27338 3/20 0.42
KDM4E B2RXH2 2/20 0.42
NPC1 O15118 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP2C19 P33261 1/20 0.41
CHRM2 P08172 1/20 0.41
HKDC1 Q2TB90 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22702081 0.83 SMN1; SMN2 (0.49) ALDH1A1SMN1; SMN2POLBMAOAMAOB
SCHEMBL22702133 0.76 ADH1B (0.46) ALDH1A1SMN1; SMN2POLBMAPTMAOA
SCHEMBL15066769 0.74 SMN1; SMN2 (0.53) ALDH1A1SMN1; SMN2POLBMAOAMAOB
SCHEMBL6866606 0.73 MAOA (0.57) ALDH1A1SMN1; SMN2POLBMAOAMAOB
SCHEMBL6866612 0.73 MAOA (0.57) ALDH1A1SMN1; SMN2POLBMAOAMAOB
SCHEMBL22307241 0.72 SMN1; SMN2 (0.47) ALDH1A1SMN1; SMN2POLBMAOAMAOB
SCHEMBL4782825 0.71 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2CYP1A2POLBCYP2D6
SCHEMBL13373201 0.70 MAOA (0.50) ALDH1A1SMN1; SMN2CYP1A2MAPTMAOA
SCHEMBL12069840 0.70 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2CYP1A2POLBCYP2D6
SCHEMBL12046092 0.70 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2CYP1A2POLBCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3319955-B1 6-AMINO-QUINOLINE-3-CARBONITRILS AS COT MODULATORS GILEAD SCIENCES INC (US) 2020-11-25 EP disclosed